somatostatin receptor agonist — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T2584	Octreotide	SMS 201-995	Somatostatin
	Octreotide (SMS 201-995) is a potent inhibitor of growth hormone, glucagon, and insulin.		Somatostatin
T28743	Seglitide acetate	MK 678,MK678,MK-678	Somatostatin
	Seglitide acetate (MK-678) is a selective agonist of sst2 somatostatin receptor.		Somatostatin
T9692	Paltusotine		Somatostatin
	Paltusotine is a nonpeptide, small molecule somatostatin type 2 (SST2) receptor agonist with high oral bioavailability. Paltusotine maintains GH and IGF-1 levels in acromegaly patients		Somatostatin
T22907	L-817,818		Others
	somatostatin sst5 receptor agonist		Others
T23073	NNC 26-9100		Others
	Somatostatin sst4 receptor agonist		Others
T27783	L-779976	L-779,976,L779,976,L779976,L 779976,L 779,976
	L-779,976 is an agonist of somatostatin receptor.
T22487	(1R,1'S,3'R/1R,1'R,3'S)-L-054,264		Others
	somatostatin sst2 receptor agonist		Others
T24860	TC-G1003	TC G1003
	TC-G1003 is an effective agonist of the somatostatin sst2 receptor.
T27787	L-797,591
	L-797,591 is a selective agonist of somatostatin receptor subtype 1.
T69836	Paltusotine HCl
	Paltusotine, also known as CRN00808, is a somatostatin receptor agonist.
TP2124	Somatostatin 1-28
	Somatostatin receptor agonist, derived from the post-translational cleavage of prosomatostatin.
T76544	Cyclic SSTR agonist octreotide
	Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .
T39207	L-803087 TFA
	L-803087 TFA is a highly potent and selective agonist of the somatostatin sst4 receptor, exhibiting a Ki value of 0.7 nM. It displays a remarkable selectivity, being over 280-fold more preferential for the sst4 receptor ...
TP2045	CH 275
	Potent somatostatin receptor 1 (sst1) agonist; displays selectivity for sst1 (IC50 values are 30.9 nM, 345 nM, > 1 μM, > 10 μM and > 10μM for human sst1, sst3, sst4, sst2 and sst5 respectively). Attenuates somatostatin r...
T11700	J-2156		Others
	The ED50 of J-2156 in rats for the relief of mechanical allodynia and mechanical hyperalgesia in the ipsilateral hindpaws was 3.7 and 8.0 mg/kg, respectively. J-2156 is a high potent, selective somatostatin receptor type...		Others
T60784	SSTR4 agonist 2
	SSTR4 agonist 2 is a potent somatostatin receptor subtype 4 (SSTR4) agonist that has the potential in SSTR4-related medical disorders research. SSTR4 pathway inhibits the processes of nociceptive and inflammatory [1].
T32511L	L-796,778 acetate	L-796,778 acetate(217480-25-6 Free base)	Somatostatin
	L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.		Somatostatin
T75248	Pasireotide (diaspartate)
	Pasireotide diaspartate (SOM230), a long-acting cyclohexapeptide and somatostatin analog, enhances agonist activity across somatostatin receptor subtypes (sst1/2/3/4/5, with pK i values of 8.2, 9.0, 9.1, <7.0, and 9.9, r...
T82883	BIM-23027
	BIM-23027 is a selective sst 2 receptor agonist (EC 50 = 0.32 nM) with effects analogous to the cyclic tetradecapeptide somatostatin (SRIF). It promotes dopamine release through a Glu-dependent mechanism [1] [2].
T35669	Neuromedin C (trifluoroacetate salt)
	Neuromedin C is a bombesin-like neuropeptide that stimulates uterine smooth muscle contraction and the release of gastrin , somatostatin, and amylase in rats. Neuromedin C is a truncated form of gastrin-releasing peptide...